Endoxifen E-isomer hydrochloride

CAS No. 1197194-61-8

Endoxifen E-isomer hydrochloride( E-Endoxifen hydrochloride )

Catalog No. M17183 CAS No. 1197194-61-8

Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
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5MG 192 In Stock
10MG 281 In Stock
25MG 448 In Stock
50MG 653 In Stock
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Biological Information

  • Product Name
    Endoxifen E-isomer hydrochloride
  • Note
    Research use only, not for human use.
  • Brief Description
    Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
  • Description
    Endoxifen, a tamoxifen metabolite, is effective specific Estrogen Response Modifier (SERM).
  • In Vitro
    Endoxifen E-isomer (1-1000 nM; 12 h) inhibits PGR gene expression in E2-induced MCF-7 cells.
  • In Vivo
    ——
  • Synonyms
    E-Endoxifen hydrochloride
  • Pathway
    Proteasome/Ubiquitin
  • Target
    Tyrosinase
  • Recptor
    ERR
  • Research Area
    Cancer
  • Indication
    ——

Chemical Information

  • CAS Number
    1197194-61-8
  • Formula Weight
    409.95
  • Molecular Formula
    C25H28ClNO2
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : ≥ 30 mg/mL. 73.18 mM
  • SMILES
    CC/C(=C(/c1ccc(cc1)O)\c1ccc(cc1)OCCNC)/c1ccccc1.Cl
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1. Chae YJ, et al. Eur J Pharmacol. 2015 Apr 5;752:1-7.
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